Opioid Receptor


Opioid receptors are a group of inhibitory G protein-coupled receptors with opioids as ligands.[1][2][3] The endogenous opioids are dynorphins, enkephalins, endorphins, endomorphins and nociceptin. The opioid receptors are ~40% identical to somatostatin receptors (SSTRs). Opioid receptors are distributed widely in the brain, and are found in the spinal cord and digestive tract.The endogenous opioid system is thought to be important in mediating complex social behaviors involved in the formation of stable, emotionally committed relationships.

  • U-54494A hydrochloride EI2837

    U-54494A hydrochloride是κ 激动剂。

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  • SDM25N hydrochloride EI2519

    SDM25N hydrochloride是活性的选择性非肽类 δ 拮抗剂。

    More
  • SB 205607 dihydrobromide EI2458

    SB 205607 dihydrobromide是选择性高亲和性非肽类δ1激动剂。

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  • Salvinorin A EI2442

    Salvinorin A是高活性的,选择性 κ 激动剂。

    More
  • Salvinorin B EI2443

    Salvinorin B是可以激活κ-opioid DREADD (KORD)。

    More
  • U-54494A hydrochloride EI2837

    U-54494A hydrochloride是κ 激动剂。

    More
  • SDM25N hydrochloride EI2519

    SDM25N hydrochloride是活性的选择性非肽类 δ 拮抗剂。

    More
  • SB 205607 dihydrobromide EI2458

    SB 205607 dihydrobromide是选择性高亲和性非肽类δ1激动剂。

    More
  • Salvinorin A EI2442

    Salvinorin A是高活性的,选择性 κ 激动剂。

    More
  • Salvinorin B EI2443

    Salvinorin B是可以激活κ-opioid DREADD (KORD)。

    More
  • U-54494A hydrochloride EI2837

    U-54494A hydrochloride是κ 激动剂。

    More
  • SDM25N hydrochloride EI2519

    SDM25N hydrochloride是活性的选择性非肽类 δ 拮抗剂。

    More
  • SB 205607 dihydrobromide EI2458

    SB 205607 dihydrobromide是选择性高亲和性非肽类δ1激动剂。

    More
  • Salvinorin A EI2442

    Salvinorin A是高活性的,选择性 κ 激动剂。

    More
  • Salvinorin B EI2443

    Salvinorin B是可以激活κ-opioid DREADD (KORD)。

    More
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